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Glucuronidation converts gemfibrozil to a potent, metabolism-dependent inhibitor of CYP2C8: implications for drug-drug interactions.
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has minor subject area list
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Alamethicin; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2C8; Dose-Response Relationship, Drug; Drug Interactions; Glucuronates; Humans; Hypolipidemic Agents; Mass Spectrometry; Microsomes, Liver; Uridine Diphosphate Glucuronic Acid
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information resource reference
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Ogilvie BW, Zhang D, Li W, Rodrigues AD, Gipson AE, Holsapple J, Toren P, Parkinson A. Glucuronidation converts gemfibrozil to a potent, metabolism-dependent inhibitor of CYP2C8: implications for drug-drug interactions. Drug Metab Dispos. 2006 Jan; 34(1):191-7.
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label
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Glucuronidation converts gemfibrozil to a potent, metabolism-dependent inhibitor of CYP2C8: implications for drug-drug interactions.
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